Hauora, Mau faaineineraa
"Esomeprazole": tohutohu mō te whakamahi, ritenga tūturu
"Esomeprazole" - he tarukino e no ki te raau taero gastrointestinal Organotropona. Te raau e antiulcer mahi, me te ko te inhibitor iraoho papu.
Te hanganga, te puka tuku "esomeprazole" tarukino
Ko wātea i roto i te puka o papa ki te inenga o te 20 me te 40 mg o kaha esomeprazole whakauru, me te rite i roto i te puka o te paura tikanga mo te otinga mō te werohanga (40 mg oko) te tarukino. papa pani, whakakorenga i e wahi i roto i te piro.
mahi pharmacological "esomeprazole" tarukino
He aha te mea te tarukino "esomeprazole"? Tohutohu mō te whakamahi whakaatu e tenei kaihoko antiulcer, e, he he turanga ngoikore, e tango te puka kaha i muri i ingestion. "Esomeprazole" inhibits te paru H + -k + -ATPase mahi, me secretion o te waikawa pūhaumāota (whakaongaongatia, basal). puta mahi e tika ana i roto i te haora i muri i ingestion o te tarukino. A, no te fariiraa i "esomeprazole" hanga ra, mo nga ra e rima, te horopeta rā tīkina - 20 mg i muri whakaongaonga mā te pentagastrin taumata mōrahi o te waikawa pūhaumāota heke te nui (e pā ana ki 90%).
Pharmacokinetics
"Esomeprazole" tohutohu mō te whakamahi ko rite te tarukino nei, ngoto i roto te tinana, tere, me te pai whenumi, herea ki pūmua tata 100% (97%). nui haere te bioavailability ki te whakamahi hia o te tarukino i 64 ki te 89%. Ko te medicament e te ahua o metabolites me excreted matua i roto i te mimi, ona he wahi iti hakari i roto i te feces.
Tuhinga "esomeprazole" teuteu
"Esomeprazole" analogues whakamahia i roto i te tūroro ki gastroesophageal mate Reflux maimoatanga me te ārai matahoki. Ko te taputapu e whakamahia ana i roto i te maimoatanga o tuwhenua o te puku duodenum ranei, mo te ārai mate puta tika ki NSAIDs.
Te raau e whakamahia ana i roto i te whewhe keté, ka pāngia duodenum puku ranei. taea te tono te reira ki tūroro kua oti nei te whakaora esophagitis, i roto i te ārai matahoki auroa. Whakaaetia tono tahi ki te tikanga "esomeprazole" raau taero antibacterial. Papa me te werohanga i roto i te therapy matatini i roto i tenei take tukua whakangaro Helicobacter pylori.
Contraindications ki te fariiraa i "esomeprazole" tarukino
Contraindications ngā tau iti iho i te tekau ma rua nga tau, ki te hypersensitivity esomeprazole, te wā o te whāngai ū. Ko te mau hopearaa o te maimoatanga tarukino kihai i i whakapumautia i roto i te hapūtanga.
Mahinga tarukino
whakamahia te raau i roto i te horopeta rā o 20-40 mg. whakaritea te roanga o te therapy te tohu talena me te fariiraa tōtika medicament "esomeprazole". Papa, me te pakeke otinga rere i iti hoki tākihi te whakamahi i te horopeta mōrahi o te 20 mg.
esophagitis Reflux Erosive tukinotia hoki wha wiki ki te horopeta rā o 40 mg. I roto i te ārai auroa o te hohokitanga i runga i te fariiraa tikanga he manawanui i roto i nei kua esophagitis i whakaorangia, kua whakaturia te horopeta ia i roto i te whānuitanga o te 20 mg.
I roto i te maimoatanga o te Reflux oesophagitis, e hāngai ana ki te whakatutuki i te tohu mate whakakaupapa, tango 20 mg o tarukino "esomeprazole". Teuteu i roto i te puka o papa, me te paura whakamahia te ki whakamatea H. Pylori, ka reira he kōrero ki te whewhe duodenal, i roto i te therapy pahekotanga - "esomeprazole" (20 mg), "Clarithromycin (500 mg)," amoxicillin "(1 g). rongoā katoa tangohia rua he ra.
mariao puku meinga e NSAIDs, e tūtohu ana ki te hamani 20 mg "esomeprazole" ia ra. Kei te whakaritea nga wa katoa te horopeta e hiahiatia ki te rata tango ki pūkete te hauora o te manawanui, te mate, te pakeke o tona akoranga, me ētahi atu āhuatanga nui.
Pānga te taha "esomeprazole" tarukino
Tūroro e tango enei taero mo te wa roa, he nui atu e pängia ana ki te hanganga o cysts glandular i roto i te kopu i te tahi atu tūroro. Ko te mau faaiteraa kino tino auau o te tinana i roto i te maimoatanga tikanga "esomeprazole" ako i runga i te tono ka tukuna he ānini me etahi tauhohe tōraro i te wahi gastrointestinal, pēnei i: kōroke, flatulence, korere, whakapairuaki, ruaki, aroaro o te mamae i roto i te puku. Na roto i te ono pānga taha ngā whakamaroke o te mucosa o te mangai, whanoke, urticaria, minamina, dermatitis. He taea Ētahi atu tauhohe, te tikanga kia pera kawea te maimoatanga i tino i raro i te mātakitaki o te mātanga.
tahi tuwhena rawa e ngoikore whānui, te whakanui ake i pā o ngā pānga taha, tae atu i runga i te wahi o te wahi kūnatu. I roto i ngā take pēnei i, whakamana maimoatanga e whakakore i te tohu o te tuwhena rawa, me te tiaki therapy. Tātari kua tata kahore pānga e hiahiatia, i reira he kahore raau.
Ara
wahine hapu "esomeprazole" analogs whakahaeretia ki te tūpato tino. kia Treatment i roto i hapūtanga kia mātakitaki i e te tākuta. whakaritea te tarukino te ki nga wahine hapu anake i roto i aua wā i reira te whai hua o ratou tinana tino nui te kino pea ki te tamaiti e parauhia te. e kore raraunga pono i runga i te pānga o te raau taero i runga i te kukune kia karo maimoatanga ki tenei rongoā ko ano, tae noa ki taea. Whakamahi o te tarukino "esomeprazole" ka rāhuitia uma-kai te.
A, no te ofatiraa o rawa te horopeta i whakaritea te ate he mōrearea ki te hauora (ki te he nui enei maumaui).
A, no te Kua tohua tohu o te manawanui tohu, pērā i hematemesis, dysphagia, whakapairuaki, whakaiti nui i roto i te taimaha tinana i roto i te wā maimoatanga "esomeprazole" i roto i te tikanga ki te whakakore whewhe tika ki te tango i te raau taero i roto i te aroaro o te mate whakapae ranei, kia mukua repara. Ki te tautuhi i te āhua mārere o te pukupuku, ko te tika ki te whakahaere i te ako.
Tūroro e whai i te kore o te sucrase-isomaltase, tuku pūāhua huahuka ātete riria mai ki whakarite "esomeprazole" taurite.
Ngā pāhekoheko "esomeprazole" ki ētahi atu taero
Ki te whakamahi tukutahi o te tarukino me "citalopram", "clomipramine", "imipramine" potentiation taea o enei āpiha, whakapai ake o te taonga kaha i roto i te toto. A, no te whakamahia i roto i te taha ki "esomeprazole" iti pai "ketoconazole" "Itraconazole" worsens ratou absorption.
A, no te whakakotahi i te "esomeprazole" ki "ATV" kua he hekenga nui i roto i te puaretanga o tenei tarukino kua. e kore te tūtohu "Esomeprazole" ako whakahaere ki te whakamahi i te wā kotahi ki te "phenytoin", "clomipramine", "imipramine" me taero pērā i "citalopram", "Diazepam", "Nelfinavir" me "Atazanavir". taea ki te ara i roto i te toto te taumata o enei taero he, na kia ai taua mea e minaminatia ki te iti o ratou pota. whakamahi te rere o «esomeprazole" me te tikanga "clarithromycin" arata'i ki te huringa nui i roto i te te rongo "esomeprazole" e tupu te whakanui ake ona e pā ana ki inhibition o pākia o te tarukino. E tika ana kia āta whakaaro instrukiyu ki te tarukino me te kōrero i te tohunga.
Ko te utu o te raau taero, arotake e pā ana ki te tarukino "esomeprazole"
riro te nuinga te tarukino i roto i te puka papa. Pharmacies "esomeprazole" taea te kitea i raro i te ingoa hokohoko "Nexium" me "Emanera". A, no te hoko koe tei te tarukino "esomeprazole" utu i runga i te horopeta o te taonga kaha i roto i tona hanganga. Ko te utu o te tarukino i te inenga o te 20 mg ( "Emanera") Ko e pā ana ki 500 moni. hoki 28 papa, me te whakaritea e te kaiwhakanao. Rongoā ki te horopeta o 40 mg o te whakauru kaha ( "Nexium" 28 papa) e taea te hokona hoki 3000 moni.
"Esomeprazole" He arotake te nuinga pai. tuhia ratou te taonga tarukino ki te tautāwhi secretion waikawa, e rua basal me whakaongaonga. Kua whakaaturia e te raau miramira tiketike i roto i te maimoatanga o ngā āhuatanga e ōrite tohu tohua i roto i te ako. I roto i therapy, tenei te tikanga i reira ko te tūponotanga iti o ngā pānga taha. Ko kore katoa ngāwari taea ki te kitea te tarukino i roto i pharmacies, etahi tūroro nei i riro "esomeprazole", te mea tiketike te utu.
Ko te hunga e ka mau te rongoā whakaritea e te tākuta i muri i te whakamāramatanga pū o te tātaritanga me te horopeta tūtohu, tohu he whakapai ake nui i roto i te hauora. Ka rite ki nga arotake, "Nexium" ko atu rongonui i roto i tūroro atu "Emanera". A, no te whakarato "Nexium" pekitīlia te ahua o te hua e hiahiatia ana i muri i pā ana ki te marama kotahi i muri i tomokanga o te therapy. Te whakapai ake ka taea e te huru puta i muri i 1.5 wiki o te maimoatanga. He tino onge pānga taha. Drug "Nexium" whai hua, e tauturu te reira ki te whakakorenga o te tikanga e whakahuatia ki roto i te tohutohu. Ko pai te hua, he mea e tika ana ki te whakaoti i te akoranga katoa, me te tino piri ki tūtohutanga o te tākuta.
Analogs "esomeprazole"
taea te kitea i te kōwhiringa e whai ake nei i analogues o te tarukino:
- "Omeprazole" - ka karanga ano "Losek", "Omez", "Ultop";
- "Rabeprazole" - he faaineineraa mohiotia i raro i te ingoa "Ontaym", "Zulbeks", "Noflyuks" "Pariet", "Hayrabezol";
- "Pantoprazole" ( "Sanpraz", "Kontrolok", "Nolpaza");
- "Lansoprazole" ( "Lanza", "Lanzoptol").
enei taero katoa i ngā pānga rite, engari rerekē ratou i ia atu i roto i to ratou uara.
Rite "esomeprazole" me "Omeprazole". E kitea rerekētanga o enei taero. "Esomeprazole" ko he poinanaha "omeprazole". Tenei faaineineraa, timata mai i te raraunga tuhinga hauora, kua he painga nui, engari he mahi rite o medicaments. "Omeprazole" Ko te uara tarukino tauanga ki te maha nui o ngā pānga taha. Ki te whakaaro tatou ki nga āhuatanga o te "esomeprazole", te aroaro te raau e rite te putanga ake o "omeprazole", te utu o e kua ngā maha tūroro. Heoi, "esomeprazole" iti iho pea ki te meinga tauhohe e hiahiatia, kia whakaaro tona hoko te atu pai atu i hoko "Omeprazole".
"Rabeprazole" me "esomeprazole" i te hanganga matū rite, hamani ratou i te mate taua. Ko tohunga whakapono e etahi mate, pērā i te mate gastroesophageal Reflux, "Rabeprazole" faaore atu tōtika, te tango i reira nga tohu pai, whai wāhi ai ki te ora tere o nga mahi pū kai. Ko te kore o te pānga pai i roto i te maimoatanga o "esomeprazole" kia pā ana ki te āhuatanga takitahi o te rauropi.
Ki te tika, whiriwhiri kia kōrero i te orotahi te tākuta. Hamani atu tahuri ki to ratou hauora, me te haere te tirohanga i roto i te wa, ka ka kia tere te ora, a ka karo koe maha pōauautanga.
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