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"Thiotriazoline": tohutohu mō te whakamahi

E takiuru koe te tarukino "Thiotriazoline"? i runga i te whakamahi o tenei aratohu rongoā ka kia whakaahuatia i roto i te taipitopito i roto i te tuhinga nei. I tua atu, ka korero ki matou a koutou e pā ana ki te puka i roto i nei te raau tomo te hoko mea, e kua e ia tohu, pānga taha me contraindications.

Ko te hanganga o te tākai tarukino me te puka tuku

I roto i te aha puka tuku medicament "Thiotriazoline"? Tohutohu ngā e te mea he maha o ngā momo rerekē. Ko te tino rongonui ko:

  • He otinga tikanga mō te werohia intramuscular me te rō-uaua. 1 ml o te kaihoko kei 0,025 g Thiotriazoline. Ano he medicament me wāhanga kōwhiringa i roto i te puka o te wai mō te werohia. E wātea ana i roto i te 4 ml ampoules (whakanohoia i roto i te kātene) te tarukino.
  • makaka "Thiotriazoline" kanohi. Na roto i te te whakamahi o te aratohu taua tikanga whakarato e 5 ml kei 50 mg o tarukino Thiotriazoline, me ētahi atu matū. Te raau e hokona i roto i nga ipu kirihou, droppers, whakanohoia i roto i te pouaka pepa.
  • "Thiotriazoline" pire. Tohutohu ki tenei puka o te tarukino whakarato e i roto i te kotahi ma papa porohita ki te mata papatahi roto 100 morfoliniymetiltriazoliltioatsetata mg, pera-ka karanga Thiotriazoline ranei. Ka rite ki atu wāhanga o te medicament mahi māngaro potato, microcrystalline cellulose, iti povidone taimaha rāpoi, konupūmā stearate me te sucrose. Ka rite ki te tikanga, i roto i te mōkihi pepa kei 50 papa.

pharmacodynamics

He aha te mea te rongoa rite "Thiotriazoline"? Tohutohu mō te Whakamahi kī e tenei tarukino antioxidant. he tika ki te antioxidant āhuatanga, antiischemic, immunomodulatory me te membrane aueue tona pai tiketike.

rongoā i Tirohia ārai whakangaromanga o hepatocytes, whai wāhi ki to ratou ora, te whakaiti i te tohu o te fatty kookuhutanga, hua i roto i te māori o te pūmua, te warowaihā, lipid me te utu ngarahu, me te whakaiti i te tūponotanga o te horapa o te necrosis tsentrolobulyarnyh te tinana pērā i te ate. I tua atu, whakapiki i tarukino kaha te wehe, me te kōtuitui o te ate, normalizes tona hanganga (matū).

Ko te āhuatanga o te tarukino

Kia pehea te kua te āhuatanga o te tarukino "Thiotriazoline"? Tohutohu mō te whakamahi o te raau taero e hiahiatia te hoki pānui. I muri i te katoa, anake i reira ka taea e koe te ako e pā ana ki te mea Whakahekea te raau taero whakaaro inhibition o tukanga oxidative i roto i te huringa Krebs, te haapa'oraa i te tahua ATP intracellular, me te whakarei ake i te whakahohenga (e vai) hāorakore glycolysis.

mōhio ana hoki e muri i tango i te taonga kaha tarukino tīmata ki te whakahohe i te pūnaha antioxidant, ngako tautāwhi i tukanga oxidative i roto i te wāhi rere pūroto o te tinana. I tua atu, whakapiki i tenei raau nga āhuatanga (rheology) o te toto e tika ana ki te faaitoitoraa o te pūnaha fibrinolytic.

Ko te āhuatanga antioxidant o te raau taero whakakitea e te meka e te hanganga o te rāpoi ngota he katote tiotrazolina whanariki, āhuatanga e te āhuatanga pitihāoratanga me te tangohāoratanga, me te hauota wānanga, e herea i te nui rawa o ngā katote hauwai.

kia mōhio hoki tatou e taea te wāhanga tarukino hohe ariu ki Radicals lipid me ngā momo hāora urupare. Ko te tika ki te āhuatanga whakaiti korerotia o te rōpū thiol tenei. I tua atu, i te medicament ārai te hanganga o ngā momo hāora urupare, taua antiradical whākōkī reactivating rite catalase, glutathione peroxidase me dismutase superoxide.

Pharmacokinetics

Ahakoa whenumi rongoā te "Thiotriazoline"? kī ako e te tarukino wā poluabsorbtsii he 30 meneti me te bioavailability - 65.5%.

tutuki mōrahi tikanga kukū toto te i roto i 1.4 haora i muri i whakahaere. e kore e Communication ki pūmua nui 10%.

I roto i ngā rahinga nui, piki te rongoā i roto i te kopa o te ate, ngakau, kopirua, kōateate me whatukuhu, me te iti - i roto i te kōpiro iti me te pūkahukahu. Thiotriazoline excreted te nuinga i nga whatukuhu.

iteraa papû

Ki te reira e taea te whakaritea ine pire, werohanga me makaka kanohi "Thiotriazoline"? i runga i te whakamahi o enei momo o ako whakaatu nga tohu e whai ake nei:

  • cirrhosis;
  • kino ate paitini, waipiro, viral, me taero (hei tauira, i muri i te fariiraa i paturopi, huaketo taero, anti-TB me te anti-puku āpiha, te whakawhānau kōrero me pōuritanga tricyclic);
  • kakā viral ma'i;
  • kakā waipiro ma'i āhua ki te mahi iti;
  • e hōloa ate fatty.

Tuhinga mō te whakamahi pata:

  • mate Corneal;
  • weranga kanohi ranei wharanga;
  • pīkaru viral.

He aha te whakamahi tonu raau ophthalmic "Thiotriazoline"? Tohutohu (Ka taea te hokona pata i tetahi whare kēmihi) ngā e te maha whakaritea tenei rongoā mo te ārai o te kanohi maroke, pūrata, me ētahi atu mate inflammatory o whekau ataata.

papa te inenga

Me pēhea e whakamahi ahau "Thiotriazoline" papa? Kei Manual mōhiohio e kia te tarukino kia tangohia roto anake. Ka rite ki te tikanga, thiotriazolin whakaritea 1 ranei 2 papa wha nga wa he ra mo te 25-30 ra.

kia te roanga o te maimoatanga ki tenei kaihoko e whakaritea e te tākuta i runga i te pūtake takitahi (i runga i te akoranga me te pakeke o te mate tīariari rānei).

Ko te otinga tarukino "Thiotriazoline": tohutohu mō te whakamahi

Werohanga "Thiotriazoline" mahi intramuscularly pâmuhia ranei. Ratou inenga whakaritea e te rata (i runga i te mate rānei). infarction myocardial me hepatitis tarukino āta patia e pâmuhia i roto i te 2 ml 2-3 wā i te ra. I roto i te cirrhosis faaterehia medicament te intramuscularly (2 ml 2-3 wā i te ra). Ko te akoranga o te maimoatanga he 60 ra.

Eye makaka "Thiotriazoline": tohutohu mō te whakamahi

Eye makaka "Thiotriazoline" Hare ki te pūwhera conjunctival. Ko te tikanga, ko te inenga mō ngā pakeke, ko te 2 pata o runga ki te 4 wā i te ra. Ki te whakaaro ki ngā tamariki, whakaritea te nui o te raau taero e anake e te tākuta tamariki. Ko te roanga o te maimoatanga me pata kanohi, a me tāuta e te rata haere.

Ka rite ki te tikanga, he kore neke atu i te 2 wiki te roanga o te maimoatanga ki tenei taputapu. Otiia ki te kitea kahore he whakapai ake te, e taea te whakawhānui ake i te akoranga ki runga ki te marama.

I roto i te take whānui pāpaka whekau ataata, me te nui, ka dropwise tua ki werohanga ocular whakahaerea (taka kē).

Hoki te ārai o whakamaroke o te kiriuhi kanohi (i te mahi i te rorohiko), me te whakamahi koe i te rongoā 2 pata i roto i te ra ki te wā o te 2 haora.

pānga taha

He aha e nga pānga taha o te tarukino e taea meinga "Thiotriazoline" (matā)? Tohutohu ki tenei tikanga kōrero e te pai noatia te tarukino ki te faatura. Heoi, mā te whakamahi i te raau taero whakaaro e taea tonu puta tauhohe koretake te.

  • pūnaha Central io: whanoke, ngoikore, waea i roto i te taringa.
  • wahi kūnatu: mangai maroke, whakapairuaki, bloating.
  • Oko me te ngakau, te pēhanga nui haere toto, tachycardia, arrhythmia, mamae ngakau.
  • pūnaha Respiratory: huangō me te hāhā o te manawa.
  • Pāwera: kirika, tauhohe hypersensitivity, angioedema.
  • tauhohe Local: whero me te mania sensation i te wāhi i werohia.
  • tauhohe Dermatological: Makere kiri, minamina, pununga honé.

Ko pata kanohi, e runga i te wahi o ratou i kitea i te pānga taha.

taunekeneke tarukino

E ai ki te tohunga, ka taea te whakamahi i te tarukino "Thiotriazoline" i roto i te taha ki te rongoa taketake tikanga mo te maimoatanga o te mate ngakau coronary. Ko e tika ana ki te meka i mea tarukino ko te kaihoko cardioprotective tenei.

Me mahara hoki käore te reira e whakaaetia te tarukino te ki te whakamahi tukutahi ki ngā rongoā e kua whakaritea ki te maimoatanga tika o te kakā etiology.

Kanohi makaka "Thiotriazoline" taea te whakaritea ki nga wahine hapu, me te i roto i te hohipera. kia hoki kia mea te reira e e whakaaetia te āhua o te hua ka mea ki te whakamahi i roto i te taha ki te tahi atu rave'a rata.

Waipiro me Drugs "Tiatriazolin" whakaū mahi tahi e te tahi o. I roto i tenei whakaaro, rāhuitia ratou te whakamahi te rere te.

Ara

Ko te hanganga ngā papa sucrose whakaaro (i roto i te nui o 2.8 mg ia papa). Ko te kupu, ki te horopeta mōrahi rā o te rongoā e taea i roto i pā ana ki 22.4 mg o te taonga. Me ki mohio tūroro, tūroro ki te mate huka mellitus tenei meka.

Ko te tikanga me wā o te rokiroki

Tino kia tiakina katoa puka "Tiatriazolin" tarukino i te marama, me te taea o ngā tamariki i te pāmahana o i 14 ki te 26 nekehanga. Ko te ora papa o te tarukino ko 3 tau.

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