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"Agapurin": tohutohu mō te whakamahi, tūturu

He aha te mea te tarukino "Agapurin"? Tohutohu mō te whakamahi, te puka tuku, me te hanganga o nga moni ka te aroaro he iti atu. I tua atu, i roto i tenei tuhinga ka ako koe e pā ana ki te take i roto i i whakaritea te tarukino te ina te tino rāhuitia tona whakamahi, ahakoa kua ia ngā pānga taha, me te pera i runga i.

Te hanganga me te ahua o te tarukino

He reira he ingoa ao i roto i te "Agapurin" tarukino? "Pentoxifylline" - ko tona ingoa tuarua tenei.

I tēnei wā e wātea ana i roto i ngā puka e rua rerekē te tarukino:

  1. pani papa Biconvex (ma), me te he i te whiti mōhinuhinu. Kei roto i tēnei raau te wāhanga kaha he pentoxifylline me matū atu (monohydrate reihuka, te kānga māngaro, colloidal silica anhydrous, talc me stearate konupora). Ki te whakaute ki te anga, ngā reira āhuatanga pērā i te konutai carmellose, tioata sucrose, paura sucrose, talc, methylparaben, Titanium hāorarua, takawai colloidal anhydrous me te hitimi.
  2. Rongoā (mārama, taekore) mo te werohia. Tenei medicament ngā pentoxifylline, konutai pūhaumāota me te wai mo te werohia.

hiahia ana ano ahau ki te whakahua i te meka e taea te kitea i te taua orotahi tarukino i roto i mekameka rongoā rite "Agapurin faataere". e ai ta ako o te tarukino i ko ia he kaihoko o te mahi auroa. Ko reira e wātea ana i roto i nga papa, e kua pani ki te paninga kiriata. Kei tēnei rongoā pentoxifylline me āhuatanga atu pērā i hypromellose, povidone, talc, me stearate konupora.

āhuatanga pharmacological

He aha te mea te tarukino "Agapurin"? kī Tohutohu mō te Whakamahi i te mea antispasmodic tenei kaihoko, me te no ki te rōpū purine. Te reira i tino whakapiki i toto tohanga, me te ona āhuatanga rheological. Ko te parau tumu whakahaere o te medicament mea he ki phosphodiesterase inhibition, me te whakanui ake i te ihirangi o ATP i erythrocytes me puni i roto i platelets ki pea matā waiwai pūngao. Nā tēnei, i roto i te vasodilation, e tukupu ana i te ātete iaia katoa (piringa), me te meneti, me te whakapiki ake i rōrahi patu kahore te huringa nui i roto i auau ngakau.

Ko te tikanga o te mahi o te tarukino

He aha te mea te huarahi o te mahi "Agapurin" tarukino? Tohutohu mō te whakamahi hoatu he whakahoki ngaio ki tenei pātai. I muri tono wewiti medicament iatuku pūngākau, a ka whakanui ake i te tuku hāora ki te oko pūkahukahu me te myocardium, he reira pānga antianginal me whakapiki i oxygenation o te toto.

Me mahara hoki käore te reira e te waihanga aroaro ahei o te whakanui ake i te āhua o te musculature romahā, i ngā o te HWM me Uaua.

A, no te rō-uaua werohia arata'i te reira ki nui haere tohanga hei utu, me te he hua i roto i te rōrahi toto e rerengia ana i roto i te-Tsu-wāhanga 1. I tua atu, tenei raau ai he hua i roto i te ihirangi o te adenosine i roto i te roro, me te he hua i runga i te mahi bioelectrical o te pūnaha io.

E ai ki te ako, ka mea he ahei o te whakaiti i te pokey o te toto, ki te whakapiki ake i te elasticity o te membrane ngeniwhero me te whakapai ake microcirculation ki te tohanga waimaero medicament.

He aha ngā āhuatanga e te rongoā "Agapurin"? Tohutohu mō te whakamahi kī e i roto i te mate occlusive matua taea (piringa) tarukino kaha arahi ki whakakorenga o cramps po i roto i te kuao kau, te tawhiti elongation o haere me te mamae i okiokinga.

Pharmacokinetics

Medicine "Agapurin" Kei te tere metabolized i roto i te ate. hua tenei metabolites kaha. Ratou kukū i roto i te rave rahi taime toto ki runga ake i te kukū o te taonga taketake.

He whakaatu aroaro medicament rite metabolites i te nui o 94%, me te toenga - i roto i te whēkau. I roto i te 4 hāora tuatahi i muri i ingestion o te raau taero tukua i roto i te nui o 90% o te toketaá whakamahia. I roto i te puka kāore i, kua whakaaturia te reira i roto i te rōrahi o te 2%. Me mahara hoki käore te reira e kore e te taonga kaha me metabolites o pentoxifylline herea ki pūmua toto.

mahi tākihi, no te waimaero decelerates metabolites putanga. Ki te kite abnormalities ate mahi roa hawhe-te ora, a ka nui haere bioavailability.

Drug "Agapurin" (papa): tohutohu mō te whakamahi

E ai ki nga tohutohu piri ki te medicament, me tangohia te reira i tetahi me te wa ano o te ra i muri i te kai i te kai, inu wai mania. Ko te tarukino i roto i tetahi take e taea ki te whakahoki ake.

inenga tuatahi o te tarukino ko 200 mg toru nga wa o te ra. Ki te waiho te manawanui he maimoatanga roa i rawakore kātakí o te tarukino ranei, ka taea te heke rite rua he horopeta kotahi, engari kia mau ki te maha o pōhiri ki.

Te tikanga e kore e inenga ia nui 1200 mg.

Na e matau ana koutou ki te whakamahi i te tarukino "Agapurin" (papa). tikanga ōrite hoki te tohutohu tono ki tuku whānui kei ngā mōhiohio e pā ana ki te taua toketaá. Heoi, ka whakamahi i te reira taea ki te whakaiti i te liunga fariiraa.

Tohutohu mō te whakamahi o te otinga mō te werohanga

Me pēhea te ki te whakamahi i te tarukino "Agapurin"? E whakaritea Papa atu pinepine atu i te rongoā injectable. Ki te hoki tetahi take e kore e taea te tango i te manawanui rongoā-waha, whakaritea ia werohanga.

Tenei faaineineraa hokona i roto i te puka otinga mō te werohanga kia whakahaerea e tetahi o nga tikanga e whai ake nei:

  1. Iv. kia diluted nga tirotiro o te ampoule i roto i te 5% otinga kūhuka i ranei i roto i 250-500 ml pūhaumāota (0.9%) te konutai pūhaumāota. kia whakahaerea āta te tarukino, e kore neke atu i 150 ml ia haora. Ki te Māna te manawanui te rongoā, whakaaetia te horopeta rā ki te whakapiki ake i runga ki te rua ampoules, ie 200 mg.
  2. Intramuscularly. whakahaere te raau i 100 mg rua he ra. e kore e waimeha te reira i te tirotiro o te oko.
  3. Intraarterially. kia tīmata Treatment o te manawanui ki te whakahaere o te ampoule kotahi, e kia kia mua-diluted i roto i te 20-50 ml o isotonic otinga konutai pūhaumāota. Ki te hiahia koe ki te therapy auroa, kia nui haere te horopeta ki 2-3 ampoules. Me diluted ratou ki 30-50 ml.

Me kï reira e takoto te nui tino arotau o te medicament aroaro te anake e te rata, a anake i roto i te akoranga o te tohutohu manawanui takitahi.

Medicament "Agapurin": tohu hoki te whakamahi

I mua i te whakamahi i tenei rongoā, kia kōrero koe tou tākuta, me te kia whakamatauria. I muri i te katoa, whakaritea rongoā te anake i raro i etahi ine. Ko te rārangi e whakaaro atu matou.

  1. disorders arataukai o te kopa e kua puta ki te puipuitua o venous rawakore microcirculation matua ranei (pērā i kaikai, tuwhenua tētere, hukapuri, a na i runga i.).
  2. disorders circulatory (piringa) i hanga nei te rite ki te hua o ngā tukanga inflammatory, atherosclerotic me te mate huka. rongoā rite whakaritea hoki claudication "taratahi", meinga nei e atherosclerosis, mate occlusive matua, me angiopathy huka.
  3. patunga rere pūroto ma'i, me te whakapeka, i te mea takenga rere pūroto. Ano, whakamahia te raau taero i roto i kaka arteriosclerosis, paresthesia, angioneyropatii, mate o Raynaud me akrozianoz.
  4. tohanga waimaero i roto i te oko o te whekau ataata (whakapeka, me te ma'i kore circulatory, iaia me te mata kiriuhi o te kanohi).
  5. State puta i muri i rere pūroto hemorrhagic ranei patu.
  6. Disorders o te taringa waenga take iaia, e kua haere tahi e rongo mate.

Contraindications ki te whakamahi o

A, no te kore e taea e koe te whakamahi i te rongoā "Agapurin"? rāhuitia te whakamahi o tenei tarukino te i raro i te tikanga me ine e whai ake nei:

  • infarction myocardial whakapeka;
  • faaite arteriosclerosis coronary kaka ranei;
  • faaite hara o manawataki ngakau;
  • porphyria;
  • hypotension matua whakakeke;
  • toto nui;
  • patu hemorrhagic whakapeka;
  • toto tuaroa;
  • hapū, uma-kai;
  • te tau o 18 tau (haumaru me te tapiri mana kihai i i whakapumautia);
  • hypersensitivity ki pentoxifylline, me ngā huānga i pārōnaki rōpū xanthine.

whakamahi tūpato o te rongoā

Ki te tiaki nui te taputapu ki te kia tono ki tūroro ki te hehema ki matua hypotension, pēhanga toto labile, kore ngakau (tonu), he haafifi i ki pakaruhanga toto, iti hoki tākihi me te ate, me ano hoki i roto i te huru i muri i te pokanga.

pānga taha

He reira tetahi ngā pānga taha i te tarukino, "Agapurin"? aratohu Papa aroaro nei ki runga ake, me te he otinga mō te werohia e taea meinga he maha o hopearaa kino. Kia whai whakaaro ano tatou ratou i roto i te kōrero atu.

  • pūnaha kūnatu: kakā cholestatic, atony intestinal, whakahōhā cholecystitis, mangai maroke me te mate o te hiahia.
  • pūnaha io: manukanuka, ohoroa, whanoke, cramps me pāhoahoa.
  • oko Toto me te kiri: huamo, whao pakarukaru, Makere kanohi, Makere te tihi o te pouaka me te mata.
  • pūnaha Cardiovascular: arrhythmia, angina teka, pectoris angina ahu whakamua, tachycardia me te pēhanga toto iti.
  • Tinana o te hematopoiesis me pūnaha hemostasis: thrombocytopenia, leukopenia, pancytopenia, gipofibrinogenemia i toto intestinal, puku, tōiti subcutaneous me kiriuhi mucous.
  • whekau rongo: kite waimaero me scotoma.
  • mate pāwera: pruritus, urticaria, angioedema , me anaphylaxis.

take o te tuwhena rawa

Eaha te tupu, ki te whakamahi koe i pota teitei te tarukino "Agapurin" (400 mg, 600 mg, 1200 mg)? I roto i tenei take, kia wheako te manawanui taua tohu pathological rite ngoikore, tohua whakaiti i roto i te pēhanga toto, whanoke, tachycardia, syncope, somnolence, te whakatakiruatanga o haurangi toniki-clonic, mate o mahara, tūāhuruiti, irritability, gastrointestinal toto tohu (hei tauira, ruaki " whenua kawhe ") me te areflexia.

I roto i tenei take titau maimoatanga symptomatic akiaki whakahaua nei i pupuri i te pēhanga toto noa, me te mahi romahā.

Motuhake tohutohu mō te whakamahi o te raau taero

He aha kia mohio koutou ki te aroaro o te whakamahi koe i te tarukino "Agapurin"? Reviews o taote titau e he pai te rongoa i tenei mahi, engari te maimoatanga e hiahia ana ratou ki te hei i raro i te mana tino o te pēhanga toto. I roto i tenei take, i roto i tūroro ki te kore te ngakau (tonu) hiahiatia te ki te whakatutuki paremata tohanga.

Me mahara hoki käore te reira e i roto i te tūroro ki te tātaritanga o "mate huka" tango taero hypoglycemic, te whakamahi o tenei kaihoko i roto i pota nui ai he suka korerotia. Na reira he tika hoki ratou whakatikatikanga whängainga.

Ki te whakamahi tukutahi o te tarukino me anticoagulants kia āta aroturuki i te huru o te pūnaha toto coagulation.

I roto i te tūroro tata nei i i pokanga, e hiahia ana koe ki te aroturuki tonu te kukū o te pūtoto, me te hematocrit.

Me heke te inenga faaterehia i roto i te tūroro ki te pēhanga toto iu iti ranei.

kia Me iwi pakeke te horopeta iti.

E ai ki ngā akoranga, e paowa tino whakaiti te miramira whakaora o te tarukino.

kia pentoxifylline hototahi ki ētahi atu rongoā e whaowhia kia tirohia i roto i te take ia takitahi.

Ngā pāhekoheko ki ētahi atu tikanga

maha whakarei ake te taonga pentoxifylline kaha te mahi o te āpiha e pā upoo- toto. Taua raau taero ngā anticoagulants hāngai, me te autaki, waikawa valproic, thrombolytics, me anitibiotiki (hei tauira, taero "Tsefamandol", "Cefoperazone", "tsefotetan").

Ka mea faarahi māngai te whai huatanga o te hypoglycemic-waha me taero antihypertensive, me te taiāki.

E kore e taea e tatou te mea e te tarukino "cimetidine" tino whakanuia ana te kukū o pentoxifylline i te toto. faarahi tenei te mōrea o ngā pānga taha.

Co-whakahaere "Agapurin" tarukino, arotake o nei e whakaaturia ana i raro nei, ki ētahi atu xanthines arata'i ki te oaoa io nui.

Methods mō te rokiroki faaineineraa, arotake o reira, te utu

Drug "Agapurin" e hokona i roto i tata nga kēmihi. Hokona 60 papa (100 mg), ka e taea ki te toharite tika i runga i 250 moni Russian koe.

Mua o tenei medicament he pai atu. Ko te aha te reira maha atu taero whakaritea ki tūroro e whai raruraru ki te oko toto.

Me mahara hoki käore te reira e te rongoā rongonui tika nui "Agapurin" i roto i te bodybuilding. bodybuilders Reviews mea e kia whakaaro tenei taputapu motuhake i te tahi atu raau taero e whakapai ake rere te toto. I muri i te katoa, ko reira te whai hua tino me ngāwari ano.

medicament Hohe i te ki te tango kaitäkaro, rite ki te hua reira e kore anake i roto i te puka o te otinga injectable, engari ano hoki i roto i te puka papa. Pharmacies tenei taputapu e taea te kitea i raro i ngā ingoa atu e tangi rite "Pentoxifylline" ranei "Trental".

kanohi te mahi matua nui haere mahi tarukino āhua o oko toto, whakaiti pokey toto , me te whakanui ake i te rere toto. Ko he ara nui ki te rave i Pumping i runga i whakangungu hākinakina, ka reira te mea he mana'o o uaua kaha mahi kutētē tenei katoa.

Whakamahia tenei rongoā kia bodybuilders ite tino tupato, no te mea e taea e meinga ngāwari reira he tuwhena rawa, me te maha o ngā pānga taha.

Kia mau ki "Agapurin" pai i roto i te pouri, wahi maroke te wahi i reira he kore whai wāhi ki ngā tamariki taitamariki. Ko te kupu pāmahana rokiroki o te tarukino, ko te 10-15 anake nekehanga. rā paunga tohua i runga i te tākai me he rua tau. I muri i tenei wā, rāhuitia whakamahi tarukino te.

I roto i te mutunga, mōhio kotahi ano e kore e waiho tatou whaiaro whakarite-ratou tango i tēnei rongoā. kia roanga o te maimoatanga me te inenga kia whakaritea e te rata mo te manawanui ngā.

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