Tikanga e tika ana "waikawa Tranexamic" ko he tarukino antifibrinolytic, mahi anti-inflammatory me antiallergic, me te pānga hemostatic korerotia ina bleedings e e pā ana ki te hua i roto i te fibrinolysis. I te matua o te tarukino ko te inhibition o plasminogen activator me plasmin inhibition o te hanganga o peptides kaha me kinins whai wāhi tika i roto i tauhohe inflammatory, me te mate pāwera. I roto i te tua, he taputapu pērā i "waikawa Tranexamic", tino e whakaroa te wa thrombin. Ki te whakaaro ki te āhuatanga pharmacokinetics o te raau taero anti-fibrinolytic i muri ingestion te riro te reira 30-50% o tona dosing tuatahi, te rawa i kitea ai nohanga wē kotahi rau - kotahi rau e waru tekau meneti i muri i te whakamahi. pānga Antifibrinolytic i roto i te kopa tiaki hoki ma rima - whitu haora, me te wē - mō te whitu waru ranei haora i muri i whakahaere o te tarukino "waikawa Tranexamic". Ko te utu o tenei taputapu ko e pā ana ki 1300 moni, a ka taea e te hoko e koe i te reira i roto i tata nga kēmihi.
hua tarukino Antifibrinolytic te i roto i te puka o papa o e rua rau me te rima tekau ranei rima rau koma haumano, hei otinga mo te werohia, me te he otinga te tikanga mo te whakahaere-waha. He pai hāngai mō te maimoatanga me te ārai o te toto katoa o te puka inenga i runga, i whakapataritari he hua i roto i te fibrinolysis whānui. Hei tauira, kaihoko tino maha whakahaere, huaina i ki rite "waikawa Tranexamic" i roto i te puku mārere o te repeure ranei taiaki, kanisā, wawaotanga hāparapara i runga i nga whekau o te pouaka, me ate mate. Kei ngā ano tango ā-o te ewe me te kulukia toto i roto i te rārangi o tohu ki te ūnga. I tua atu, te whakamahi tarukino "waikawa Tranexamic" pau o haematuria, angioedema, dermatitis mate pāwera, katoatia, paitini, me te tarukino hikaka, pununga honé. I tua atu, tohua tenei tarukino te mo te pharyngitis kaha, laryngitis, tonsillitis, stomatitis, nasal, uterine me te puku toto, niho tango i roto i tūroro pāngia ki hemorrhagic diathesis. Ka rite ki te pai ki te taputapu pērā i "waikawa Tranexamic", me marama, i tua atu i copious.
Ko te tono motuhake, me te dosing rongoā, e whakatakotoria takitahi ratou i roto i ia take, e hāngai ana i runga i te āhuatanga haumanu homai. Heoi, ka rite ki te tikanga, i te wa whakaaetia te ki te tango i ki kaua e neke atu i te 1-1.5 karamu. I roto i tenei take, te whakamahi o te liunga lahi ko e rua ki te wha nga wa he ra, me te roanga o te maimoatanga - i toru ki te rima ra. horopeta Single mō te whakahaere rō-uaua ko te 10-15 mg / kg.
Ko te contraindications matua ki te whakamahi o tenei taputapu ko nga tikanga pērā i toto subarachnoid, thromboembolism, täkihi, tirohanga tae waimaero, me Thrombosis venous hohonu. I tua atu, e kore koutou e te whakamahi i tenei rongoā i roto i te take o te hypersensitivity takitahi hapū ranei. pānga te taha e pā ana ki te rōpū o āpiha anti-fibrinolytic, whakakitea rite whanoke, sleepiness, hypotension, tachycardia, ngoikore, me te mamae pouaka.