HauoraMau faaineineraa

"Metoprolol": arotake, tohu hoki te whakamahi, te ako me te analogues

He aha te mahi e hiahia ana ahau rongoā "Metoprolol"? Mua o tenei faaineineraa, e te aroaro ona momo tuku, hanganga, me ngā pānga taha i raro. korero hoki matou ki a koutou e pā ana ki te mea he contra-tohu me te raau taero, i roto i te mea horopeta kia tangohia reira, ki te reira e te tahi atu analogues.

Ko te hanganga o te tarukino me ona puka tuku

I roto i te mea puka hokona te rongoā "Metoprolol"? Mua mea e taea te kitea te rongoā e toru ngā momo o te tarukino. A feruri i te take o te puka, me te hanganga i roto i te kōrero atu.

  • Papa. Kei te reira i te wāhanga hohe pērā i metoprolol tartrate (100, 50, me te 25 milligrams). I tua atu, Kei te medicament wāhanga ngaahi houalotú, me te anhydrous takawai colloidal, cellulose microcrystalline, te konutai carboxymethylstarch (momo A) me te stearate konupora. I roto i te hoko o te medicament riro papa 50, 10, 30, 20 40 ranei ia mōkihi.
  • Papa ki ngā āhuatanga tuku ukauka ( "succinate metoprolol") papa pani. Kei roto ratou rite matū kaha me excipients. I roto i te pharmacies taea te kitea taua rongoā i te 30, 20 ranei 10 papa ia mōkihi.
  • Ko te otinga mō werohanga rō-uaua i roto i ampoules o 5 ml. I roto i te hoko o te tarukino mai i roto i te pouaka kātene o 10 oko.

Ko te āhuatanga pharmacological o te tarukino

He aha te tikanga o te rongoā "Metoprolol"? Ka kia te aroaro Tuhinga mo te whakamahi o te taputapu i raro. Na e hiahia ana ahau ki te korero ki a koutou e pā ana ki te mea he āhuatanga pharmacological o te tarukino.

Ka mea no rongoā ki te blockers beta-adrenergic cardioselective. e kore e whakaatu te reira i ngā āhuatanga membrane aueue me e kore mahi sympathomimetic ā-. Heoi, ko te tarukino kaha ko te antihypertensive, antiarrhythmic me te kaihoko antianginal.

Ko te ahei o te whakaiti i te auau o te auau ngakau o te manawanui te medicament, whakaiti contractility myocardial me excitability, puhoi AV-āriponga, me te whakaiti i tono hāora myocardial.

Ka rite ki te tikanga, kitea te pānga antihypertensive i roto i te tūroro i muri noa ra tekau ma wha i muri i tango i te raau taero. Ko te medicament whakaiti te auau o te whakaeke ki tachycardia supraventricular, angina pectoris me te fibrillation Atrial. Ka rite ki te hua, manawataki ngakau noa o te manawanui.

Papa ki tuku whakaroa ( "succinate metoprolol") i te painga nui i runga i tikanga. tukua ratou ki a koe te pupuri i te kukū tamau o te huānga kaha i roto i te toto, reira whakarato i te pānga haumanu pai puta noa i te ra. Me mahara hoki käore te reira e te mahi o "succinate Metoprolol" āwhina ki te whakaiti i te mōrea o te bradycardia me ngoikore, ki te whānuitanga iti, pānga nga uaua maeneene o te bronchi.

Pharmacokinetics (absorption, pākia me excretion o te tarukino)

Mō te tohu mō te whakamahi lekarstvai whakaahua i raro ngā "Metoprolol" analogues tarukino, engari inaianei kia kōrero a pā ana ki te āhuatanga pharmacokinetic.

Tenei te tikanga rawa hohoro a tata rawa (e pā ana ki 95%) whenumi te. Kei te nuinga o te wā tae kukū wē mōrahi i muri i 50-110 meneti i muri i ingestion.

Ko te tono tuatahi o te bioavailability tarukino ko 50%. Toutou faarahi te reira ki te 70%. E te ara, e faarahi te kohi o kai te bioavailability o te raau taero i te 20-40%. reira e faarahi hoki, ki te he ate cirrhosis te manawanui. Communication ki pūmua i runga i toharite 10%.

Ka mea ô i pai medicament te placental me toto-roro tauārai. Hoki i roto i ngā rahinga iti, tu te reira i roto i, me te ki te waiu uma.

metabolized te raau i roto i te ate. Na whai metabolites mahi pharmacological. Mō 5% o te Agent excreted e nga whatukuhu tonu. Therapy Kātaki ki mahi tākihi iti titau whakaiti atu horopeta ako ranei. Heoi, kia pōturi iho pākia o taero raruraru i roto i te ate mahi. I roto i tenei take, kia heke te inenga.

Rongoā "Metoprolol": tohu hoki te whakamahi

He he rawa te rārangi nui o ngā āhuatanga pathological i e whakahaerea te tarukino te. Kia titiro tatou ki a ratou.

  • akathisia, i meinga e antipsychotics;
  • takawhita matua o te 1 me te tohu 2 matua takawhita (pea monotherapy, a i roto i ngā take kino - me Diuretics me ētahi atu taero antihypertensive);
  • thyrotoxicosis (he wahi anake o te maimoatanga matatini);
  • ārai o whakaeke angina me angina;
  • prophylaxis o migraine;
  • takahi o te manawataki cardiac (hei tauira, arrhythmia, me tachycardia supraventricular paroxysmal, tachycardia supraventricular);
  • ki te whakaiti i te mōrea o te tahuti nei, me te tahumaero i roto i te mate Cardiovascular me te mate te AVC;
  • ārai tuarua o infarction myocardial me whakapeka infarction myocardial;
  • prolapse takirere mitral;
  • Ko idiopathic cardiomyopathy Dilated;
  • giperkinez Cardiovascular Tino, hyperkinetic syndrome cardiac, disorders o te ngakau.

Reviews o medicament

E ai ki nga arotake o te hunga e kua tonu kua tuku ki te tarukino, i te reira tōtika akakoromaki i te mahi, me te pānga pai i runga i te ngakau. Heoi, kia tuhia te reira e pahono te tahi mau tūroro ki rongoa kore e tino pai. Ka rite ki te tikanga, he tika ki te meka e te mea he maha contraindications me ngā pānga taha tenei. Ko te take i roto i ngā tūroro amuamu, whakaahua i raro i runga i te taenga o nga moni.

Contraindications ki te whakamahi o te rongoā

Na, inaianei e mohio ana koe he aha te tikanga te tarukino "Metoprolol" (tohu mō te whakamahi i whakaahuatia tika i runga). Heoi, i tenei tarukino he maha o contraindications kua. Ko ētahi o ēnei:

  • ātete takitahi (i.e. hypersensitivity ki wāhanga kaha ngaahi houalotú ranei);
  • atrioventricular 2 poraka, me te tohu 3;
  • whakamahi kotahi-wā ki inhibitors Mao;
  • pā sinuauricular;
  • Ua faaite disorders circulatory (piringa);
  • pakohu bradycardia (auau ngakau, ki te - i te iti rawa e ono tekau ia meneti);
  • e suka me ahua labile o te mate huka;
  • syndrome pakohu mate;
  • manawanui aro ki bronchospasm (i.e., huangō arahau, me te whakautu nui arahau);
  • acidosis pūkoro;
  • hypotension (iti iho i te 100 mm HG ..);
  • ru cardiogenic (kore te te tarukino tūtohutia mō ngā tūroro ki te tātaritanga o "infarction myocardial whakapeka" ranei whakapae ki reira);
  • kore whakapeka ngakau, ma'i (atamira 2, me te 3), me te uncompensated.

Rāhuitanga i runga i te whakamahi o te tarukino (fariiraa ki te tūpato tino)

I roto i te aha kia iti take ki te fariiraa "Metoprolol" tarukino? tohunga Reviews mea e ki kia heke te horopeta o medicament i hyperthyroidism, emphysema, hītori mate pāwera, huangō arahau, Bronchitis kore-mate pāwera, psoriasis, pheochromocytoma, disorders ate, whatukuhu, me te (i ētahi wā), korekore, gravis myasthenia me te rehunga whānui.

He mea taea ki te hoatu tamariki rongoā "Metoprolol"? rāhuitia te whakamahi o tenei rongoā e tangata i raro i te 18 tau o te tau te. He kanga i runga i moni te fariiraa toro ki hapu wahine me te u,. Kore ki te ū ki enei tūtohutanga, i reira te mea he mōrearea nui o bradycardia, suka, me hypotension i roto i te aiû fanau apî.

Ki te hiahia koe i te horopeta o rongoā i roto i te whāngai ū, i roto i tenei wa o te hohipera kia mutu.

Drugs "Metoprolol" me "succinate Metoprolol": tohutohu mō te whakamahi

Tikanga, te medicament "metoprolol" tango i te ra i roto i te nui o 100 mg. Ai mea kua wehea rōrahi ki te maha pota. I roto i te tikanga ki te whakatutuki i te pānga haumanu pai, e taea te nui haere te fariiraa i te 2 ngā wā. Heoi, e kore e nui ake te horopeta mōrahi o te tarukino 400 mg.

A, no te whakahaere kotahi-wā werohia rō-uaua i 2 ki te 5 mg o te faaineineraa. I roto i tenei take, te inenga mōrahi ko 15-20 mg. I roto i te ngaro o te pānga e hiahiatia ana whakaaetia ki anō-tomo i te taonga tarukino (i roto i te 5 meneti).

Whakakore i te whakarite o te tarukino kia kia āta. Ko te tikanga i meatia tenei te hoki nga ra kotahi tekau i raro i te te tirotiro motuhake o te tākuta.

inenga tuatahi o te tarukino "succinate metoprolol" ki tachycardia supraventricular, pectoris angina, arrythmia me takawhita ko e pā ana ki 50-100 mg kotahi te ra. A, no te tiaki therapy o infarction myocardial te fariiraa i medicament i roto i te horopeta o 200 mg.

Ko te roanga iti o te maimoatanga tikanga "metoprolol succinate" Ko 3 marama. Ki te pāngia te manawanui kei ki te kore te ngakau ma'i, whakaritea te inenga te takitahi. Tuatahi, tangohia te raau taero i roto i te nui o 12.5 mg kotahi ia mo 2 wiki, a ka nga ra 14, rererua te horopeta te.

I kātakí āhua pai o te medicament ai tona horomanga mōrahi ia ra tae 200 mg.

pānga te taha. mua

Ka taea e kino te reira i te rongoā tinana "Metoprolol"? Reviews o tenei faaineineraa kei te rota o te mōhiohio e muri i tona whakauru i reira he nunu'a kovi. Mō nei i roto i te pātai i te ari?

  • Mai i te pūnaha io: uaua ngoikore, rohirohi, ri'ari'ai, korekore, pāhoahoa, manukanuka, tērā o te nekeneke me te hinengaro tauhohe, heke whakarongo, paresthesia i te topito, waimaero mahara wā-poto, te momoe ranei, hei kōrero, ohoroa.
  • Mai i te rongo: te secretion iti o te wai roimata, heke kite, pīkaru, te mamae, me te maroke kiriuhi mucous o nga kanohi, waea i roto i te taringa.
  • pūnaha manawa-iaia: arrhythmia, pakohu bradycardia, angina teka, raruraru āriponga infarction, e tukupu ana te pēhanga toto, he faaiteraa o vasospasm, hypotension orthostatic, heke contractility myocardial me te whanoke.
  • Mai i te pūnaha kūnatu: mangai maroke, mamae puku, whakapairuaki, mahi ate rerekē, kōroke, ruaki, korere, me ngā huringa i roto i te reka.
  • Kiri: minamina, alopecia reversible, hikaka, Makere, hikaka, sweating, exacerbation o psoriasis, photodermatosis, exanthema me psoriasiform kiri tauhohe.
  • pūnaha Respiratory: hāhā o manawa, popoketanga nasal, bronchospasm me te uaua exhaling.
  • I runga i te wahi o te pūnaha endocrine: hypothyroidism, e suka me Hyperglycemia.
  • Whakamātau Laboratory: thrombocytopenia, agranulocytosis, hyperbilirubinemia, leukopenia, me whākōkī ate mā'olunga.
  • Ko te pānga i runga i te kukune o te wahine hapu i raro i tono: intrauterine retardation tupu, bradycardia me te e suka.

I tua atu, i muri i te fariiraa i raau mea pūrongo etahi tūroro te takanga o te mamae tahi mamae hoki ranei. iwi whakaatu tino onge e kua paku nui haere ratou papatipu tinana, heke libido mananga ranei.

arata'iraa Motuhake i runga i te whakamahi o te raau taero

Na i roto i tetahi rongoā ka taea e koe te hoko i te tarukino "Metoprolol". E kore te te tohutaka e hiahiatia ana. Heoi, no te tūroro tango rongoā kia aroturuki auau i te rata te rongoā. Ko rawa pono hoki te hunga tūroro e pāngia mate huka angina ranei tenei.

Kei te mohio te reira e na roto i te whakanui ake i te inenga (neke atu i te 200 mg ia ra) heke cardioselective. I roto i te aroaro o te kore ngakau therapy tīmata te i muri i anake tae te wā utu te.

Iwi e whakamahi arotahi whakapā, me whakaaro koutou e i roto i te horopaki o te maimoatanga, "metoprolol" production iti o roimata inu.

I te tahi taime i tenei kopare rongoā etahi tohu o hyperthyroidism. I roto i tenei withdrawal ohorere o te tarukino i roto i ngā tūroro ki te mate mea te contraindicated, mai e haamaitai te reira i te tohu.

Ki te tika, te mahi te manawanui kia mōhio tonu te anesthesiologist ki therapy tarukino.

I roto i te maimoatanga, te whakapōauau, "metoprolol" he tika ki te kakahu e tika ana. Ko e tika ana ki te meka e kia meinga i te tarukino tauhohe mate pāwera ki te kiri e tika ana ki te rongo ki te rā tenei.

E kore e taea e tatou te mea e te rongoā "Metoprolol" (analogues o tenei rongoā i roto i ngā) i roto i te paari e taea meinga te ahua o te whakanui ake i bradycardia, tohua whakaiti i roto i te pēhanga toto, poraka atrioventricular. Ko enei tūroro titau aha mana motuhake.

I tua atu, i roto i te maimoatanga ki tenei raau kia pehi i peia he waka, me te aukati i ngā akomanga ngā mahi mōrearea e rapua e kukū tiketike me tauhohe tere whakamātau tinana. Kei te tūtohu hoki te reira e te whakauru o te waihā.

Ngā analogs tarukino

He aha te ki te taea ki te hoko i te rongoā whakaritea e te tākuta, "metoprolol" te manawanui ko te? E wātea ana ona analogues i roto i tetahi rongoā. Te nuinga o ratou i roto i te taonga kaha rite, ko te kupu kua reira te taua āhuatanga rite tarukino mea. I roto i enei kia whakahuatia te raau taero e whai ake nei: "Acre Metoprolol", "Metolol", "Metokor Adifarm" me etahi atu.

I muri i te rironga raraunga tikanga ki te manawanui tohutohu ki tirohia ki nga tohutohu piri, me ki kōrero ki te tākuta. Ko tenei e tika ana ki te meka e kia rerekē te tikanga te whiwhi i te toketaá tikanga i runga ake.

He aha atu e tenei analogs rongoā? Whakakapia taea tikanga whakarite o te tākuta hei te rongoā e whai ake nei: "bisoprolol" "Metoprolol-Ratiopharm", "Metokard", "Korvitol", "Metozok", "Lidalok", "Serdol", "Egilok", "Emzok" me etahi atu.

Me pēhea te ki te rokiroki me te te nui rongoā?

Na e matau ana koutou he aha te tikanga te, pehea me i roto i te aha te inenga ki te tango i rongoā "Metoprolol". Rokiroki i te reira i roto i te wahi raumati (hei tauira, i roto i te pouaka) ranei he ruma i reira e kore e te pāmahana nui 25 nekehanga. I roto i tenei take, kia tiakina te tarukino i te rā tika.

Pa'epa'e ora o te tarukino mea me te nuinga o ona ritenga i o e rima nga tau i te rā o te production. I muri i tenei wā, rāhuitia te rongoā e whakamahia ana i roto i ngā take whakaora, me te prophylactic te. kia whiua te reira.

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